Litcius/Paper detail

PFKFB3 inhibitors as potential anticancer agents: Mechanisms of action, current developments, and structure-activity relationships

Yinhu Wang, Chen Qu, Tingting Liu, Chunhui Wang

2020European Journal of Medicinal Chemistry74 citationsDOIOpen Access PDF

Topics & Concepts

Allosteric regulationChemistryGlycolysisPhosphofructokinase 2Activator (genetics)EnzymeCancer cellBiochemistryWarburg effectPhosphofructokinaseFructose 2,6-bisphosphateKinaseCancerBiologyReceptorGeneticsCancer, Hypoxia, and MetabolismATP Synthase and ATPases ResearchMitochondrial Function and Pathology