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Access to azonanes <i>via</i> Pd-catalyzed decarboxylative [5 + 4] cycloaddition with exclusive regioselectivity

Ying Liu, Yicheng He, Yang Liu, Kun Wei, Wusheng Guo

2021Organic Chemistry Frontiers33 citationsDOI

Abstract

An efficient approach for the synthesis of azonanes via Pd-catalyzed decarboxylative [5 + 4] cycloaddition has been developed. The reactions feature wide functional group tolerance with exclusive regioselectivity.

Topics & Concepts

RegioselectivityCycloadditionChemistryFunctional groupCatalysisCombinatorial chemistryOrganic chemistryPolymerCatalytic C–H Functionalization MethodsCatalytic Alkyne ReactionsCyclopropane Reaction Mechanisms