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Discovery of novel BCL6-Targeting PROTACs with effective antitumor activities against DLBCL in vitro and in vivo

Dazhao Mi, Li Cheng, Yuzhan Li, Mingyue Yao, Yan Li, Keyu Hong, Chengying Xie, Yihua Chen

2024European Journal of Medicinal Chemistry26 citationsDOIOpen Access PDF

Topics & Concepts

BCL6LymphomaChemistryCancer researchIn vivoIn vitroCarcinogenesisB cellImmunologyBiologyBiochemistryGeneticsGeneGerminal centerAntibodyProtein Degradation and InhibitorsUbiquitin and proteasome pathwaysMultiple Myeloma Research and Treatments
Discovery of novel BCL6-Targeting PROTACs with effective antitumor activities against DLBCL in vitro and in vivo | Litcius