ML162 derivatives incorporating a naphthoquinone unit as ferroptosis/apoptosis inducers: Design, synthesis, anti-cancer activity, and drug-resistance reversal evaluation
Furong Ma, Yulong Li, Maohua Cai, Wenyan Yang, Zumei Wu, Jinyun Dong, Jiang‐Jiang Qin
Topics & Concepts
ApoptosisGPX4ChemistryCancer cellProgrammed cell deathGlutathioneCell biologyBiochemistryPharmacologyCancerGlutathione peroxidaseBiologyEnzymeGeneticsFerroptosis and cancer prognosisDrug Transport and Resistance MechanismsCancer Mechanisms and Therapy