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Evaluation of PNU-159682 antibody drug conjugates (ADCs)

Dane Holte, Joseph P. Lyssikatos, Amanda Valdiosera, Zachary Swinney, Vikram Sisodiya, Joseph Sandoval, Christina Lee, Monette Aujay, Robert Tchelepi, Omar Hamdy, Christine Gu, Baiwei Lin, Hetal Sarvaiya, Marybeth A. Pysz, Amy Laysang, Samuel A. Williams, Dong Jun Lee, Magda K. Holda, James W. Purcell, Julia Gavrilyuk

2020Bioorganic & Medicinal Chemistry Letters24 citationsDOI

Topics & Concepts

LinkerChemistryConjugateDrugCombinatorial chemistryAnthracyclineMetaboliteStereochemistrySmall moleculeMechanism of actionIn vivoDrug discoveryPharmacologyBiochemistryIn vitroBiologyInternal medicineCancerComputer scienceMathematicsOperating systemMedicineBiotechnologyBreast cancerMathematical analysisHER2/EGFR in Cancer ResearchMonoclonal and Polyclonal Antibodies ResearchChronic Lymphocytic Leukemia Research
Evaluation of PNU-159682 antibody drug conjugates (ADCs) | Litcius