Novel 1H-pyrazolo[3,4-d]pyrimidin-6-amino derivatives as potent selective Janus kinase 3 (JAK3) inhibitors. Evaluation of their improved effect for the treatment of rheumatoid arthritis
Yuan Yin, Chengjuan Chen, Ru-Nan Yu, Lei Shu, Zhijian Wang, Tiantai Zhang, Dayong Zhang
Topics & Concepts
ChemistryRheumatoid arthritisJanus kinase 3TofacitinibJanus kinasePharmacologyArthritisKinaseIn vivoBiochemistryIn vitroImmunologyMedicineBiologyBiotechnologyCytotoxic T cellAntigen-presenting cellCytokine Signaling Pathways and InteractionsRheumatoid Arthritis Research and TherapiesMyeloproliferative Neoplasms: Diagnosis and Treatment