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Indomethacin-based PROTACs as pan-coronavirus antiviral agents

Jenny Desantis, Beatrice Mercorelli, Marta Celegato, Federico Croci, Alessandro Bazzacco, Massimo Baroni, Lydia Siragusa, Gabriele Cruciani, Arianna Loregian, Laura Goracci

2021European Journal of Medicinal Chemistry93 citationsDOIOpen Access PDF

Topics & Concepts

Vero cellDrug discoveryCoronavirusChemistryBiologyVirologyVirusBiochemistryCoronavirus disease 2019 (COVID-19)MedicinePathologyDiseaseInfectious disease (medical specialty)Protein Degradation and InhibitorsPeptidase Inhibition and AnalysisCAR-T cell therapy research
Indomethacin-based PROTACs as pan-coronavirus antiviral agents | Litcius