A sensitive HPLC-FLD method for the quantification of alpelisib, a novel phosphatidylinositol 3-kinase inhibitor, in rat plasma: Drug metabolism and pharmacokinetic evaluation in vitro and in vivo
Seong-Wook Seo, Ji‐Min Kim, Dong-Gyun Han, Dongho Geum, Hwayoung Yun, In‐Soo Yoon
Topics & Concepts
PharmacokineticsChemistryIn vivoPharmacologyBioanalysisBioavailabilityHigh-performance liquid chromatographyChromatographyOral administrationClinical chemistryMedicineBiochemistryBiotechnologyBiologyToxin Mechanisms and ImmunotoxinsPI3K/AKT/mTOR signaling in cancerChronic Lymphocytic Leukemia Research