Discovery of chalcone analogues as novel NLRP3 inflammasome inhibitors with potent anti-inflammation activities
Cheng Zhang, Yue Hu, Ping Sun, Lei Hua, Shuli Liang, Yitao Ou, Dan Wu, Xinyi Wu, Hao Chen, Ying Hao, Wenhui Hu, Zhongjin Yang
Topics & Concepts
InflammasomeChemistryChalconeInflammationPharmacologyLead compoundBiochemistryIn vitroStereochemistryReceptorImmunologyBiologyInflammasome and immune disordersMacrophage Migration Inhibitory FactorCholesterol and Lipid Metabolism