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Discovery of disubstituted xylylene derivatives as small molecule direct inhibitors of Keap1-Nrf2 protein-protein interaction

Dhulfiqar Ali Abed, Sumi Lee, Longqin Hu

2020Bioorganic & Medicinal Chemistry27 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryPotencyKEAP1XylyleneOxidative stressDrug discoveryDocking (animal)BiochemistryLead compoundReactive oxygen speciesPharmacologyDrugSmall moleculeIn vitroCombinatorial chemistryTranscription factorOrganic chemistryGeneNursingMedicineGenomics, phytochemicals, and oxidative stressGlutathione Transferases and PolymorphismsRedox biology and oxidative stress
Discovery of disubstituted xylylene derivatives as small molecule direct inhibitors of Keap1-Nrf2 protein-protein interaction | Litcius