SAR based in-vitro anticholinesterase and molecular docking studies of nitrogenous progesterone derivatives
Muafia Jabeen Amin, Ghulam Abbas Miana, Umer Rashid, Khondaker Miraz Rahman, Hidayatullah Khan, Abdul Sadiq
Topics & Concepts
ButyrylcholinesteraseAcetylcholinesteraseDocking (animal)AchéChemistryIC50CholinergicGalantamineCholinesteraseInhibitory postsynaptic potentialEnzymePharmacologyIn vitroActive siteDonepezilBiochemistryInternal medicineDiseaseBiologyMedicineNursingDementiaCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsPhosphodiesterase function and regulation