A role for BET proteins in regulating basal, dopamine-induced and cAMP/PKA-dependent transcription in rat striatal neurons
Jace Jones-Tabah, Ryan D. Martin, Jennifer J. Chen, Jason C. Tanny, Paul B.S. Clarke, Terence E. Hébert
Topics & Concepts
BRD4BromodomainCell biologyTranscription factorGene knockdownTranscription (linguistics)BET inhibitorHistoneChemistryPromoterRegulation of gene expressionEffectorG protein-coupled receptorEnhancerBiologyNuclear proteinTranscriptional regulationGene expressionNucleosomePhosphorylationSignal transductionStriatumProtein kinase ANucleus accumbensG proteinNuclear export signalNuclear transportKinaseMolecular biologyDopamineProtein Degradation and InhibitorsClick Chemistry and ApplicationsChromatin Remodeling and Cancer