Investigation of the inhibitory activity of triterpenoids isolated from Actinidia polygama stems against β-glucuronidase via enzyme kinetics, molecular docking, and molecular dynamics analyses
Nguyen Viet Phong, Myungsook Heo, Le Ba Vinh, Young Ho Kim, Seo Young Yang
Topics & Concepts
ChemistryActinidiaGlucuronidaseKineticsEnzymeEnzyme kineticsDocking (animal)TriterpenoidMolecular dynamicsBiochemistryStereochemistryBotanyComputational chemistryActive sitePhysicsNursingQuantum mechanicsBiologyMedicinePharmacological Effects of Natural CompoundsNatural product bioactivities and synthesisNatural Antidiabetic Agents Studies