Design, synthesis, and tumor drug resistance reversal activity of novel hederagenin derivatives modified by nitrogen-containing heterocycles
Wentao Huang, Yingjie Wang, Si Xu, Hui Qiao, Haoran Cheng, Linxu Wang, Shuqi Liu, Qingjian Tian, Ruodong Wang, Hongbo Wang, Yi Bi
Topics & Concepts
ChemistryMultiple drug resistancePaclitaxelIn vivoP-glycoproteinCisplatinPharmacologyRhodamine 123In vitroEffluxMitoxantroneStereochemistryCancerBiochemistryChemotherapyInternal medicineMedicineAntibioticsBiologyBiotechnologyNatural product bioactivities and synthesisPhytochemical compounds biological activitiesToxin Mechanisms and Immunotoxins