Synthesis and evaluation of ursolic acid-based 1,2,4-triazolo[1,5-a]pyrimidines derivatives as anti-inflammatory agents
Tianyi Zhang, Chunshi Li, Ping Li, Xueqian Bai, Shu-Ying Guo, Ying Jin, Shengjun Piao
Topics & Concepts
Ursolic acidChemistryCelecoxibIn vitroAnti-inflammatoryCyclooxygenasePharmacologyNitric oxideDocking (animal)EnzymeOxadiazoleBiochemistryMedicineOrganic chemistryChromatographyNursingSynthesis and biological activitySynthesis and Biological EvaluationQuinazolinone synthesis and applications