Litcius/Paper detail

β-Lactam antibiotic targets and resistance mechanisms: from covalent inhibitors to substrates

Montserrat Mora-Ochomogo, Christopher T. Lohans

2021RSC Medicinal Chemistry228 citationsDOIOpen Access PDF

Abstract

Overview of β-lactam antibiotics and the proteins with which they covalently interact, focusing on penicillin-binding proteins and serine β-lactamases.

Topics & Concepts

AntibioticsCovalent bondAntibiotic resistanceChemistryMicrobiologyBiologyBiochemistryOrganic chemistryAntibiotic Resistance in BacteriaAntibiotics Pharmacokinetics and EfficacyPneumocystis jirovecii pneumonia detection and treatment