Repurposing of antitumor drug candidate Quisinostat lead to novel spirocyclic antimalarial agents
Ruoxi Li, Dazheng Ling, Tongke Tang, Zhenghui Huang, Manjiong Wang, Fei Mao, Jin Zhu, Lubin Jiang, Jian Li, Xiaokang Li
Topics & Concepts
Plasmodium falciparumPharmacologyDrugCytotoxicityDrug repositioningMalariaAntimalarial AgentChemistryHistone deacetylaseBiologyBiochemistryIn vitroImmunologyHistoneGeneHIV/AIDS drug development and treatmentMalaria Research and ControlCholinesterase and Neurodegenerative Diseases