Design, synthesis, and antitumor activity of benzimidazole derivatives as CDK4/6 inhibitors
Xiu Jun Wang, Xiao Hou, Luyao Zhang, Bing-Yan Wang, Mingyu Wu, Huijie Chen, Wentao Jiang, Yue Qiao, Meng-xin Lu, Hui-Hui Hao, Ting Geng, Jing-Ting Qin, Jing Ji, Bin Liu, Ping Wei
Topics & Concepts
BenzimidazoleChemistryHeLaCytotoxicityIC50Docking (animal)MTT assayCell cultureStereochemistryCell cycleCell growthCancer researchPharmacologyCellIn vitroBiochemistryBiologyOrganic chemistryNursingMedicineGeneticsAdvanced Breast Cancer TherapiesHER2/EGFR in Cancer ResearchCancer therapeutics and mechanisms