Evaluation of In Vitro Models for Assessment of Human Intestinal Metabolism in Drug Discovery
Mari Davies, Prabha Peramuhendige, Lloyd King, Melanie Golding, Apoorva Kotian, Mark Penney, Syeda A.B. Shah, Nenad Manevski, Nenad Manevski
Topics & Concepts
EnterocyteSulfationChemistryIn vitroMetaboliteMetabolismIntestinal mucosaDrug metabolismMicrosomeIntestinal epitheliumBiochemistrySmall intestineBiologyEpitheliumInternal medicineGeneticsMedicinePharmacogenetics and Drug MetabolismAnalytical Chemistry and ChromatographyDrug Transport and Resistance Mechanisms