A synthesis of a rationally designed inhibitor of cytochrome P450 8B1, a therapeutic target to treat obesity
Eunhee Chung, Samuel D. Offei, U-Ter Aondo Jia, Juan C. Estévez, Yessenia Perez, Hadi D. Arman, Francis K. Yoshimoto
Topics & Concepts
Cytochrome P450Cholic acidCYP3A4ChemistryEndocrinologyPharmacologyInternal medicineObesityCholesterolBiochemistryMetabolismMedicinePharmacogenetics and Drug MetabolismDrug Transport and Resistance MechanismsInflammatory mediators and NSAID effects