In silico study of 1-benzoyl-3-methylthiourea derivatives activity as epidermal growth factor receptor (EGFR) tyrosine kinase inhibitor candidates
Ruswanto Ruswanto, Amir Musadad Miftah, Daryono Hadi Tjahjono, Siswandono
Topics & Concepts
ErlotinibEpidermal growth factor receptorIn silicoThioureaChemistryTyrosine kinasePharmacologyDrugEGFR inhibitorsBioavailabilityReceptor tyrosine kinaseCarcinogenDocking (animal)Tyrosine-kinase inhibitorReceptorBiochemistryCancerBiologyMedicineInternal medicineOrganic chemistryNursingGeneSynthesis and biological activityComputational Drug Discovery MethodsCancer therapeutics and mechanisms