Discovery of compounds that reactivate p53 mutants in vitro and in vivo
Geetha Durairaj, Özlem Demir, Bryant Lim, Roberta Baronio, Delia F. Tifrea, Linda Hall, Jacob C. DeForest, Linda Lauinger, Maryam M.J. Fallatah, Clinton Yu, Hosung Bae, Dawei Lin, Jin Kwang Kim, Faezeh Salehi, Cholsoon Jang, Feng Qiao, Richard H. Lathrop, Lan Huang, Robert A. Edwards, Scott D. Rychnovsky, Rommie E. Amaro, Peter Kaiser
Topics & Concepts
In vivoIn vitroMutantChemistryComputational biologyPharmacologyBiologyBiochemistryGeneticsGeneCancer-related Molecular PathwaysCancer Research and TreatmentsUbiquitin and proteasome pathways