Synthesis, computational and experimental pharmacological studies for (thio)ether-triazine 5-HT6R ligands with noticeable action on AChE/BChE and chalcogen-dependent intrinsic activity in search for new class of drugs against Alzheimer's disease
Kinga Czarnota-Łydka, Sylwia Sudoł-Tałaj, Katarzyna Kucwaj‐Brysz, Rafał Kurczab, Grzegorz Satała, Modesto de Candia, Francesco Samarelli, Cosimo Altomare, Alessia Carocci, Alexia Barbarossa, Ewa Żesławska, Monika Głuch‐Lutwin, Barbara Mordyl, Monika Kubacka, Natalia Wilczyńska-Zawal, Magdalena Jastrzębska‐Więsek, Anna Partyka, Nadia Khan, Małgorzata Więcek, Wojciech Nitek, Ewelina Honkisz-Orzechowska, Gniewomir Latacz, Anna Wesołowska, Antonio Carrieri, Jadwiga Handzlik
Topics & Concepts
ChemistryThio-Biological activityStereochemistryAgonistReceptorIn vitroBiochemistrySynthesis and Characterization of Heterocyclic CompoundsSynthesis and biological activityChemical Reaction Mechanisms