Radiosynthesis and initial preclinical evaluation of [11C]AZD1283 as a potential P2Y12R PET radiotracer
Isaac M. Jackson, Pablo J. Buccino, E. Carmen Azevedo, Mackenzie Carlson, Audrey Luo, Emily M Deal, Mausam Kalita, Samantha T. Reyes, Xia Shao, Corinne Beinat, Sydney C. Nagy, Aisling M. Chaney, David Anders, Peter J. H. Scott, Mark A. Smith, Bin Shen, Michelle L. James
Topics & Concepts
In vivoMicrogliaRadiosynthesisNeuroinflammationPositron emission tomographyChemistryRadioligandContext (archaeology)Preclinical imagingPharmacologyIn vitroMolecular imagingBiochemistryNuclear medicineMedicineImmunologyBiologyInflammationPaleontologyBiotechnologyNeuroinflammation and Neurodegeneration MechanismsAdenosine and Purinergic SignalingTryptophan and brain disorders