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Integration of a microfluidic multicellular coculture array with machine learning analysis to predict adverse cutaneous drug reactions

Lor Huai Chong, Terry Ching, Hui Jia Farm, Gianluca Grenci, Keng‐Hwee Chiam, Yi‐Chin Toh

2022Lab on a Chip28 citationsDOI

Abstract

model achieves an average of 87.5% accuracy (correct prediction rate), 75% specificity (prediction rate of true negative drugs), and 100% sensitivity (prediction rate of true positive drugs). We then employ the MCA and the SVM training algorithm to prospectively identify the skin-sensitizing likelihood and mechanism-of-action for obeticholic acid (OCA), a farnesoid X receptor (FXR) agonist which has undergone clinical trials for non-alcoholic steatohepatitis (NASH) with well-documented cutaneous side effects.

Topics & Concepts

Multicellular organismMicrofluidicsDrug reactionDrugNanotechnologyComputer scienceChemistryComputational biologyBiologyPharmacologyMaterials scienceCellBiochemistryBiosimilars and Bioanalytical MethodsAdvancements in Transdermal Drug DeliveryMonoclonal and Polyclonal Antibodies Research
Integration of a microfluidic multicellular coculture array with machine learning analysis to predict adverse cutaneous drug reactions | Litcius