Structural basis of tolvaptan binding to the vasopressin V2 receptor
Hongli Liu, Haiyang Zhong, Yixiao Zhang, Hua-rui Xue, Zhengshuo Zhang, Kequan Fu, Xudong Cao, Xiao-chun Xiong, Dong Guo
Topics & Concepts
TolvaptanVasopressin receptorAutosomal dominant polycystic kidney diseaseChemistryVasopressinArginine vasopressin receptor 2AntagonistComputational biologyMolecular dynamicsReceptorBiophysicsMedicineKidneyBiologyInternal medicineBiochemistryComputational chemistryGenetic and Kidney Cyst DiseasesCircadian rhythm and melatoninIon Transport and Channel Regulation