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Structure and dynamics in drug discovery

Haixin Wei, J. Andrew McCammon

2024npj Drug Discovery.58 citationsDOIOpen Access PDF

Abstract

The roles of computing in structure-based drug discovery are considered, from early studies based on some of the first experimental structures of enzyme-inhibitor complexes, through the use of advanced molecular dynamics simulations and machine learning methods. This perspective aims to explore the history, current trends, and future directions of these methodologies.

Topics & Concepts

DrugDrug discoveryDynamics (music)Computer scienceMedicinePsychologyPharmacologyBioinformaticsBiologyPedagogyComputational Drug Discovery MethodsProtein Structure and DynamicsPharmacogenetics and Drug Metabolism
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