Litcius/Paper detail

Design and characterization of cereblon-mediated androgen receptor proteolysis-targeting chimeras

Akshay D. Takwale, Seunghyun Jo, Yeong Uk Jeon, Hyung Soo Kim, Choong Hoon Shin, Heung Kyoung Lee, Sunjoo Ahn, Chong Ock Lee, Jae Du Ha, Jeong‐Hoon Kim, Jong Yeon Hwang

2020European Journal of Medicinal Chemistry72 citationsDOI

Topics & Concepts

CereblonAndrogen receptorChemistryLNCaPIn vivoProteolysisProtein degradationProstate cancerProteasomeCancer researchReceptorUbiquitinCell biologyBiochemistryUbiquitin ligaseCancerInternal medicineBiologyMedicineBiotechnologyEnzymeGeneProtein Degradation and InhibitorsMultiple Myeloma Research and TreatmentsPeptidase Inhibition and Analysis