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Molecular basis for regulation of the class I phosphoinositide 3-kinases (PI3Ks), and their targeting in human disease

Alexandria L Shaw, Isobel Barlow-Busch, John E. Burke

2025Biochimica et Biophysica Acta (BBA) - Molecular and Cell Biology of Lipids8 citationsDOI

Topics & Concepts

Phosphoinositide 3-kinaseAllosteric regulationCell biologyBiologyRegulatorSignal transductionPI3K/AKT/mTOR pathwayChemotaxisChemistryCD74GeneComputational biologyTyrosine kinaseClass (philosophy)SignallingP110αReceptorProtein subunitReceptor tyrosine kinaseRegulation of gene expressionKinaseCell signalingPlasma protein bindingGeneticsPhosphatidylinositolJurkat cellsPI3K/AKT/mTOR signaling in cancerChronic Lymphocytic Leukemia ResearchMetabolism, Diabetes, and Cancer
Molecular basis for regulation of the class I phosphoinositide 3-kinases (PI3Ks), and their targeting in human disease | Litcius