Discovery of novel benzofuro[3,2-b]quinoline derivatives as dual CDK2/Topo I inhibitors
Yaoguang Huang, Wenwu Liu, Shuoqi Huang, Deping Li, Chang Xu, Xiaowen Jiang, Mingyue Liu, Xin Liu, Chengze Zhu, Limeng Wu, Huanhua Chen, Zihua Xu, Qingchun Zhao
Topics & Concepts
Cyclin-dependent kinase 2ChemistryQuinolineCell cycleTopoisomeraseRegulatorApoptosisKinaseCell growthCyclin-dependent kinase 1Cancer researchBiochemistryEnzymeBiologyOrganic chemistryGeneCancer therapeutics and mechanismsSynthesis and bioactivity of alkaloidsCancer Mechanisms and Therapy