Litcius/Paper detail

Straightforward Access to Thiocyanates via Dealkylative Cyanation of Sulfoxides

Uroš Todorović, Immo Klose, Nuno Maulide

2021Organic Letters16 citationsDOIOpen Access PDF

Abstract

Thiocyanates, versatile building blocks in organic synthesis, are shown to be easily accessible via an interrupted Pummerer reaction of sulfoxides. This facile dealkylative functionalization proceeds under mild conditions through electrophilic activation of the sulfoxide partner. The resulting thiocyanate itself can serve as a handle for diversification in a straightforward one-pot procedure.

Topics & Concepts

ChemistryElectrophileSulfoxideCyanationCombinatorial chemistryThiocyanateSurface modificationOrganic chemistryCatalysisPhysical chemistrySulfur-Based Synthesis TechniquesChemical Synthesis and ReactionsCatalytic C–H Functionalization Methods