Modified bile acids and androstanes—Novel promising inhibitors of human cytochrome P450 17A1
Yaraslau Dzichenka, Michail Shapira, Aliaksei Yantsevich, Tatsiana Cherkesova, Ljubica Grbović, Marina P. Savić, Sergey A. Usanov, Suzana Jovanović-Šanta
Topics & Concepts
CYP17A1SteroidEnzymeChemistryCytochrome P450Bile acidHydroxylationIn silicoAndrostaneSide chainStereochemistryBiochemistryHormoneOrganic chemistryGenePolymerPharmacogenetics and Drug MetabolismHormonal Regulation and HypertensionEstrogen and related hormone effects