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Design, synthesis, and biological evaluation of novel pyrido-dipyrimidines as dual topoisomerase II/FLT3 inhibitors in leukemia cells

Mohamed A. Abdelgawad, Fatma El Zahraa Ammar Mohamed, Phoebe F. Lamie, Syed Nasir Abbas Bukhari, Mohammad M. Al‐Sanea, Arafa Musa, Mohammed Elmowafy, AbdElAziz A. Nayl, Ahmed Karam Farag, Sameeha M. Ali, Mohamed E. Shaker, Hany A. Omar, Mohammed K. Abdelhameid, Manal M. Kandeel

2022Bioorganic Chemistry12 citationsDOI

Topics & Concepts

AmsacrineTopoisomeraseChemistryApoptosisAnnexinLeukemiaCell cultureIn vitroHL60EnzymeMolecular biologyBiochemistryBiologyImmunologyGeneticsCancer therapeutics and mechanismsLung Cancer Research StudiesAcute Lymphoblastic Leukemia research
Design, synthesis, and biological evaluation of novel pyrido-dipyrimidines as dual topoisomerase II/FLT3 inhibitors in leukemia cells | Litcius