Endogenous vitamin E metabolites mediate allosteric PPARγ activation with unprecedented co-regulatory interactions
Sabine Willems, Leonie Gellrich, A. Chaikuad, Stefan Kluge, Oliver Werz, Jan Heering, Stefan Knapp, Stefan Lorkowski, Manfred Schubert‐Zsilavecz, Daniel Merk
Topics & Concepts
Allosteric regulationPeroxisome proliferator-activated receptorRegulatorChemistryPeroxisomeAllosteric modulatorNuclear receptorAgonistBiochemistryCell biologyReceptorPPAR agonistPharmacologyMediatorTranscription factorBiologyGenePeroxisome Proliferator-Activated ReceptorsAdipose Tissue and MetabolismGenomics, phytochemicals, and oxidative stress