Synthesis and anticancer evaluation of 6-azacyclonol-2,4,6-trimethylpyridin-3-ol derivatives: M3 muscarinic acetylcholine receptor-mediated anticancer activity of a cyclohexyl derivative in androgen-refractory prostate cancer
Ujjwala Karmacharya, Prakash Chaudhary, Dongchul Lim, Sadan Dahal, Bhuwan Prasad Awasthi, Hee Dong Park, Jung‐Ae Kim, Byeong‐Seon Jeong
Topics & Concepts
DU145ChemistryMuscarinic acetylcholine receptorPharmacologyCancer cellAgonistLNCaPCancer researchBiochemistryReceptorCancerInternal medicineBiologyMedicineReceptor Mechanisms and SignalingPharmacogenetics and Drug MetabolismInflammatory mediators and NSAID effects