Inhibition of human and rat placental 3β-hydroxysteroid dehydrogenase/Δ5,4-isomerase activities by insecticides and fungicides: Mode action by docking analysis
Jingjing Li, Fuhong Tian, Yunbing Tang, Lei Shi, Shaowei Wang, Zhiyan Hu, Yang Zhu, Yiyan Wang, Huitao Li, Ren‐Shan Ge, Xiaoheng Li
Topics & Concepts
PregnenoloneChemistryTriclosanNon-competitive inhibitionUncompetitive inhibitorTributyltinIC50EnzymeBiochemistryNAD+ kinasePharmacologySteroidBiologyIn vitroHormoneMedicineOrganic chemistryPathologyEstrogen and related hormone effectsEffects and risks of endocrine disrupting chemicalsHormonal Regulation and Hypertension