Systematic comparison of competitive and allosteric kinase inhibitors reveals common structural characteristics
Huabin Hu, Oliver Laufkötter, Filip Miljković, Jürgen Bajorath
Topics & Concepts
Allosteric regulationChemistryKinaseEnzymeNon-competitive inhibitionAllosteric enzymeSmall moleculeComputational biologyBiochemistryBiologyComputational Drug Discovery MethodsProtein Structure and DynamicsMicrobial Natural Products and Biosynthesis