Synthesis and preliminary evaluation of 211At-labeled inhibitors of prostate-specific membrane antigen for targeted alpha particle therapy of prostate cancer
Ganesan Vaidyanathan, Ronnie C. Mease, Il Minn, Jae‐Yeon Choi, Ying Chen, Hassan M. Shallal, Choong Mo Kang, Darryl McDougald, Vivek Kumar, Martin G. Pomper, Michael R. Zalutsky
Topics & Concepts
In vivoBiodistributionProstate cancerGlutamate carboxypeptidase IIChemistryRadionuclide therapyPotencyDOTAProstateLigand (biochemistry)In vitroLipophilicityCancerCancer researchPharmacologyBiochemistryMedicineReceptorInternal medicineBiologyBiotechnologyRadiopharmaceutical Chemistry and ApplicationsProstate Cancer Treatment and ResearchPeptidase Inhibition and Analysis