Absolute membrane protein abundance of P-glycoprotein, breast cancer resistance protein, and multidrug resistance proteins in term human placenta tissue and commonly used cell systems: Application in physiologically based pharmacokinetic modeling of placental drug disposition
Zubida M. Al‐Majdoub, Jolien J. M. Freriksen, Angela Colbers, Jeroen van den Heuvel, Jan J. Koenderink, Khaled Abduljalil, Brahim Achour, Jill Barber, Rick Greupink, Amin Rostami‐Hodjegan
Topics & Concepts
Physiologically based pharmacokinetic modellingPlacentaHuman placentaDispositionChemistryDrugPharmacologyAbundance (ecology)Fetal membranePharmacokineticsCellBiochemistryBiologyPregnancyFetusGeneticsPsychologyFisherySocial psychologyPregnancy and Medication ImpactPharmacological Effects and Toxicity StudiesDrug Transport and Resistance Mechanisms