In Vitro Characterization of Ertugliflozin Metabolism by UDP-Glucuronosyltransferase and Cytochrome P450 Enzymes
Kimberly Lapham, Ernesto Callegari, Julie Cianfrogna, Jian Lin, Mark Niosi, Christine C. Orozco, Raman Sharma, Theunis C. Goosen
Topics & Concepts
GlucuronidationChemistryMetabolismUGT2B7Cytochrome P450EnzymeMicrosomeBiochemistryPharmacogenetics and Drug MetabolismDrug Transport and Resistance MechanismsMetabolism, Diabetes, and Cancer