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Conjugation of a Blood Brain Barrier Peptide Shuttle to an Fc Domain for Brain Delivery of Therapeutic Biomolecules

Marco Cavaco, Silvia Frutos, Paula Oliete, Javier Valle, David Andreu, Miguel A. R. B. Castanho, Miquel Vila‐Perelló, Vera Neves

2021ACS Medicinal Chemistry Letters30 citationsDOIOpen Access PDF

Abstract

). Overall, we demonstrated the potential of Fc-PepH3 as a versatile platform readily adaptable to diverse drugs of therapeutic value to treat different brain conditions.

Topics & Concepts

Blood–brain barrierBiomoleculePeptideBrain diseaseNeuroscienceComputational biologyComputer scienceChemistryNanotechnologyMedicineBiochemistryMaterials scienceBiologyCentral nervous systemPathologyDiseaseRNA Interference and Gene DeliveryMonoclonal and Polyclonal Antibodies ResearchNanoparticle-Based Drug Delivery
Conjugation of a Blood Brain Barrier Peptide Shuttle to an Fc Domain for Brain Delivery of Therapeutic Biomolecules | Litcius