Sulfonamide-based 4-anilinoquinoline derivatives as novel dual Aurora kinase (AURKA/B) inhibitors: Synthesis, biological evaluation and in silico insights
Mohammad M. Al‐Sanea, Ahmed Elkamhawy, Sora Paik, Kyeong Lee, Ahmed M. El Kerdawy, Bukhari Syed Nasir Abbas, Eun Joo Roh, Wagdy M. Eldehna, Heba A.H. Elshemy, Rania B. Bakr, Ibrahim Ali Farahat, Abdulaziz Ibrahim Alzarea, Sami I. Alzarea, Khalid Saad Alharbi, Mohamed A. Abdelgawad
Topics & Concepts
ChemistryAurora kinaseDruggabilitySulfonamideKinaseStereochemistryDocking (animal)QuinolineIn silicoIC50BiochemistryCancer researchCellIn vitroCell cycleBiologyMedicineOrganic chemistryNursingGeneMicrotubule and mitosis dynamicsCancer-related Molecular PathwaysPhotosynthetic Processes and Mechanisms