Litcius/Paper detail

Sulfonamide-based 4-anilinoquinoline derivatives as novel dual Aurora kinase (AURKA/B) inhibitors: Synthesis, biological evaluation and in silico insights

Mohammad M. Al‐Sanea, Ahmed Elkamhawy, Sora Paik, Kyeong Lee, Ahmed M. El Kerdawy, Bukhari Syed Nasir Abbas, Eun Joo Roh, Wagdy M. Eldehna, Heba A.H. Elshemy, Rania B. Bakr, Ibrahim Ali Farahat, Abdulaziz Ibrahim Alzarea, Sami I. Alzarea, Khalid Saad Alharbi, Mohamed A. Abdelgawad

2020Bioorganic & Medicinal Chemistry44 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryAurora kinaseDruggabilitySulfonamideKinaseStereochemistryDocking (animal)QuinolineIn silicoIC50BiochemistryCancer researchCellIn vitroCell cycleBiologyMedicineOrganic chemistryNursingGeneMicrotubule and mitosis dynamicsCancer-related Molecular PathwaysPhotosynthetic Processes and Mechanisms