Structural basis of sphingosine-1-phosphate receptor 1 activation and biased agonism
Zhenmei Xu, Tatsuya Ikuta, Kouki Kawakami, Ryoji Kise, Qian Yu, Ruixue Xia, Mingxia Sun, Anqi Zhang, Changyou Guo, Xuehui Cai, Zhiwei Huang, Asuka Inoue, Yuanzheng He
Topics & Concepts
AgonismSphingosineSphingosine-1-phosphateReceptorFunctional selectivityChemistrySphingosine-1-phosphate receptorG protein-coupled receptorCell biologySignal transductionComputational biologyNeuroscienceBiochemistryBiologyPolitical scienceLawPoliticsSphingolipid Metabolism and SignalingReceptor Mechanisms and SignalingLipid Membrane Structure and Behavior