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Epigenetic BET reader inhibitor apabetalone (RVX-208) counters proinflammatory aortic gene expression in a diet induced obesity mouse model and in human endothelial cells

Sylwia Wasiak, Laura Tsujikawa, Emily Daze, Dean Gilham, Stephanie C. Stotz, Brooke D. Rakai, Chris Sarsons, Li Fu, Salman Azhar, Ravi Jahagirdar, Michael Sweeney, Jan O. Johansson, Norman C.W. Wong, Ewelina Kulikowski

2022Atherosclerosis18 citationsDOI

Topics & Concepts

Proinflammatory cytokineInflammationBromodomainEndocrinologyInternal medicineEndothelial dysfunctionInsulin resistanceMedicineBiologyDiabetes mellitusImmunologyEpigeneticsBiochemistryGeneProtein Degradation and InhibitorsClick Chemistry and ApplicationsAdipose Tissue and Metabolism
Epigenetic BET reader inhibitor apabetalone (RVX-208) counters proinflammatory aortic gene expression in a diet induced obesity mouse model and in human endothelial cells | Litcius