Epigenetic BET reader inhibitor apabetalone (RVX-208) counters proinflammatory aortic gene expression in a diet induced obesity mouse model and in human endothelial cells
Sylwia Wasiak, Laura Tsujikawa, Emily Daze, Dean Gilham, Stephanie C. Stotz, Brooke D. Rakai, Chris Sarsons, Li Fu, Salman Azhar, Ravi Jahagirdar, Michael Sweeney, Jan O. Johansson, Norman C.W. Wong, Ewelina Kulikowski
Topics & Concepts
Proinflammatory cytokineInflammationBromodomainEndocrinologyInternal medicineEndothelial dysfunctionInsulin resistanceMedicineBiologyDiabetes mellitusImmunologyEpigeneticsBiochemistryGeneProtein Degradation and InhibitorsClick Chemistry and ApplicationsAdipose Tissue and Metabolism