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Rational design and optimization of acylthioureas as novel potent influenza virus non-nucleoside polymerase inhibitors

Xinjin Liu, Zhichao Xu, Jinsen Liang, Ting Xu, Wenting Zou, Lijun Zhu, Yihe Wu, Chune Dong, Ke Lan, Shuwen Wu, Hai‐Bing Zhou, Hai‐Bing Zhou

2023European Journal of Medicinal Chemistry11 citationsDOI

Topics & Concepts

VirusDruggabilityInfluenza A virusNucleosideVirologyChemistryFavipiravirIn vivoPolymeraseAntiviral drugRational designIn vitroOrthomyxoviridaePharmacologyBiologyEnzymeBiochemistryMedicineGeneCoronavirus disease 2019 (COVID-19)BiotechnologyInfectious disease (medical specialty)DiseasePathologyGeneticsInfluenza Virus Research Studiesinterferon and immune responsesViral Infections and Immunology Research
Rational design and optimization of acylthioureas as novel potent influenza virus non-nucleoside polymerase inhibitors | Litcius