Discovery of novel BTK PROTACs for B-Cell lymphomas
Yunpeng Zhao, Yongzhi Shu, Jun Lin, Zhendong Chen, Qiong Xie, Yanning Bao, Lixue Lu, Nannan Sun, Yonghui Wang
Topics & Concepts
Bruton's tyrosine kinaseChemistryTyrosine kinaseIbrutinibMutantCovalent bondCancer researchBiochemistryBiologySignal transductionChronic lymphocytic leukemiaImmunologyGeneLeukemiaOrganic chemistryProtein Degradation and InhibitorsChronic Lymphocytic Leukemia ResearchMultiple Myeloma Research and Treatments