A detailed computational study on binding of kinase inhibitors into β-cyclodextrin: inclusion complex formation
Maryam Faraj Pour Mojdehi, Mokhtar Ganjali Koli, Mahsa Dolatkhah Ouch Bolagh, Mina Ghane Gardeh, Seyed Majid Hashemianzadeh
Abstract
It is well known that the limited aqueous solubility of some drugs often reduces their bioavailability to targets.
Topics & Concepts
CyclodextrinInclusion (mineral)ChemistryCombinatorial chemistryBiochemistryMineralogyComputational Drug Discovery MethodsDrug Solubulity and Delivery SystemsEnzyme Structure and Function