A New Paroxetine-Based GRK2 Inhibitor Reduces Internalization of the μ-Opioid Receptor
Renee A. Bouley, Zara Y. Weinberg, Helen V. Waldschmidt, Yu‐Chen Yen, Scott D. Larsen, Manojkumar A. Puthenveedu, J.J.G. Tesmer
Topics & Concepts
InternalizationBeta adrenergic receptor kinaseG protein-coupled receptor kinaseG protein-coupled receptorKinomePharmacologyAgonistChemistryKinaseReceptorBiologyBiochemistryReceptor Mechanisms and SignalingNeuropeptides and Animal PhysiologyProtein Kinase Regulation and GTPase Signaling