Discovery of new piperaquine hybrid analogs linked by triazolopyrimidine and pyrazolopyrimidine scaffolds with antiplasmodial and transmission blocking activities
Lívia M. Feitosa, Rodolfo Rodrigo F. França, M.De L. Ferreira, Anna Caroline Campos Aguiar, Guilherme de Souza, Sarah El Chamy Maluf, Juliana Oliveira de Souza, Luana Carlos Campisano Zapata, Denise Duarte, Inês Morais, Fátima Nogueira, Maria Cristina Nonato, Luiz C. S. Pinheiro, Rafael V. C. Guido, Núbia Boechat
Topics & Concepts
ChemistryPyrimidineStereochemistryQuinolineCombinatorial chemistryOrganic chemistryTuberculosis Research and EpidemiologyQuinazolinone synthesis and applicationsMalaria Research and Control