Design, synthesis, biological evaluation of 6-(2-amino-1H-benzo[d]imidazole-6-yl)quinazolin-4(3H)-one derivatives as novel anticancer agents with Aurora kinase inhibition
Chengcheng Fan, Ting Zhong, Huarong Yang, Ying Yang, Daoping Wang, Xiaosheng Yang, Yongnan Xu, Yanhua Fan
Topics & Concepts
Aurora kinaseChemistryKinaseAurora inhibitorAurora A kinaseCytotoxicityIC50Aurora B kinaseCancer cellProtein kinase AApoptosisCancer researchBiochemistryCell cycleCellCancerIn vitroBiologySpindle apparatusGeneticsCell divisionMicrotubule and mitosis dynamicsCancer-related Molecular PathwaysPhotosynthetic Processes and Mechanisms